Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_02312
Ion Channel
Potassium voltage-gated channel subfamily A member 1
Peptide Function
Blocker
Gene Name
KCNA1
Activity Data (nM)
IC50
2 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GVPINVSCTGSPQCIKPCKDAGMRFGKCMNRKCHCTPK
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
Atto488-agitoxin 2
Peptide Species
Leiurus hebraeus (Hebrew deathstalker scorpion) (Leiurus quinquestriatus hebraeus)
Peptide Name
Potassium channel toxin alpha-KTx 3.2
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−90 mV
Temperature
18–22 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available